7ue1: Difference between revisions

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'''Unreleased structure'''


The entry 7ue1 is ON HOLD
==HIV-1 Integrase Catalytic Core Domain Mutant (KGD) in Complex with Inhibitor GRL-142==
<StructureSection load='7ue1' size='340' side='right'caption='[[7ue1]], [[Resolution|resolution]] 3.00&Aring;' scene=''>
== Structural highlights ==
<table><tr><td colspan='2'>[[7ue1]] is a 2 chain structure with sequence from [https://en.wikipedia.org/wiki/Human_immunodeficiency_virus_1 Human immunodeficiency virus 1]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=7UE1 OCA]. For a <b>guided tour on the structure components</b> use [https://proteopedia.org/fgij/fg.htm?mol=7UE1 FirstGlance]. <br>
</td></tr><tr id='method'><td class="sblockLbl"><b>[[Empirical_models|Method:]]</b></td><td class="sblockDat" id="methodDat">X-ray diffraction, [[Resolution|Resolution]] 3&#8491;</td></tr>
<tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat" id="ligandDat"><scene name='pdbligand=7OA:(3S,3aR,5R,7aS,8S)-hexahydro-4H-3,5-methanofuro[2,3-b]pyran-8-yl+[(2S,3R)-4-[{[2-(cyclopropylamino)-1,3-benzothiazol-6-yl]sulfonyl}(2-methylpropyl)amino]-1-(3,5-difluorophenyl)-3-hydroxybutan-2-yl]carbamate'>7OA</scene>, <scene name='pdbligand=SO4:SULFATE+ION'>SO4</scene></td></tr>
<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[https://proteopedia.org/fgij/fg.htm?mol=7ue1 FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=7ue1 OCA], [https://pdbe.org/7ue1 PDBe], [https://www.rcsb.org/pdb/explore.do?structureId=7ue1 RCSB], [https://www.ebi.ac.uk/pdbsum/7ue1 PDBsum], [https://prosat.h-its.org/prosat/prosatexe?pdbcode=7ue1 ProSAT]</span></td></tr>
</table>
== Function ==
[https://www.uniprot.org/uniprot/Q9YUI7_9HIV1 Q9YUI7_9HIV1]


Authors: Aoki, M., Aoki-Ogata, H., Bulut, H., Hayashi, H., Davis, D., Hasegawa, K., Yarchoan, R., Ghosh, A.K., Pau, A.K., Mitsuya, H.
==See Also==
 
*[[Retroviral integrase 3D structures|Retroviral integrase 3D structures]]
Description: HIV-1 Integrase Catalytic Core Domain Mutant (KGD) in Complex with Inhibitor GRL-142
__TOC__
[[Category: Unreleased Structures]]
</StructureSection>
[[Category: Hayashi, H]]
[[Category: Human immunodeficiency virus 1]]
[[Category: Pau, A.K]]
[[Category: Large Structures]]
[[Category: Ghosh, A.K]]
[[Category: Aoki M]]
[[Category: Aoki, M]]
[[Category: Aoki-Ogata H]]
[[Category: Hasegawa, K]]
[[Category: Bulut H]]
[[Category: Mitsuya, H]]
[[Category: Davis D]]
[[Category: Aoki-Ogata, H]]
[[Category: Ghosh AK]]
[[Category: Bulut, H]]
[[Category: Hasegawa K]]
[[Category: Davis, D]]
[[Category: Hayashi H]]
[[Category: Yarchoan, R]]
[[Category: Mitsuya H]]
[[Category: Pau AK]]
[[Category: Yarchoan R]]