Lapatinib: Difference between revisions

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New page: ===Pharmacokinetics=== {| class="wikitable" border="1" width="40%" style="text-align:center" |- ! colspan="6" align="center"| Glitazone [[Pharmaceutical_Drugs#Pharmacokinetics_Translated...
 
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{| class="wikitable" border="1" width="40%" style="text-align:center"
{| class="wikitable" border="1" width="40%" style="text-align:center"
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!  colspan="6" align="center"| Glitazone [[Pharmaceutical_Drugs#Pharmacokinetics_Translated|Pharmacokinetics]] Comparison at Equivalent Dosages <ref>doi: 10.1111/j.1365-2125.2007.02986.x</ref><ref>PMID:18997160</ref><ref>PMID: 9454824</ref><ref>PMID: 17594391</ref>
!  colspan="6" align="center"| Glitazone [[Pharmaceutical_Drugs#Pharmacokinetics_Translated|Pharmacokinetics]] <ref>PMC:2679105</ref>
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! Parameter
! Parameter
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! [[Pharmaceutical_Drugs#Tmax|T<sub>max</sub>]] (hr)  
! [[Pharmaceutical_Drugs#Tmax|T<sub>max</sub>]] (hr)  
! Lapatinib (Tykerb)
! 4
! Sunitinib (Sutent)
! Sunitinib (Sutent)
! Sorafenib (Nexavar)
! Sorafenib (Nexavar)
|-
|-
! [[Pharmaceutical_Drugs#Cmax|C<sub>max</sub>]] (ng/ml)  
! [[Pharmaceutical_Drugs#Cmax|C<sub>max</sub>]] (ng/ml)  
! Lapatinib (Tykerb)
! 115
! Sunitinib (Sutent)
! Sunitinib (Sutent)
! Sorafenib (Nexavar)
! Sorafenib (Nexavar)
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! [[Pharmaceutical_Drugs#Half_Life_.28T1.2F2.29|T<sub>1/2</sub>]] (hr)
! [[Pharmaceutical_Drugs#Half_Life_.28T1.2F2.29|T<sub>1/2</sub>]] (hr)
! Lapatinib (Tykerb)
! 9.6
! Sunitinib (Sutent)
! Sunitinib (Sutent)
! Sorafenib (Nexavar)
! Sorafenib (Nexavar)
|-
|-
! [[Pharmaceutical_Drugs#Area_Under_the_Curve_.28AUC.29|AUC]] (ng/ml/hr)
! [[Pharmaceutical_Drugs#Area_Under_the_Curve_.28AUC.29|AUC]] (ng/ml/hr)
! Lapatinib (Tykerb)
! 1429
! Sunitinib (Sutent)
! Sunitinib (Sutent)
! Sorafenib (Nexavar)
! Sorafenib (Nexavar)
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! Sorafenib (Nexavar)
! Sorafenib (Nexavar)
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|-
! Clearance (ml/hr)
! Dosage (mg)
! Lapatinib (Tykerb)
! 100
! Sunitinib (Sutent)
! Sorafenib (Nexavar)
|-
! Equivalent Dosage (mg)
! Lapatinib (Tykerb)
! Sunitinib (Sutent)
! Sunitinib (Sutent)
! Sorafenib (Nexavar)
! Sorafenib (Nexavar)