3pvu: Difference between revisions

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[[Image:3pvu.jpg|left|200px]]
[[Image:3pvu.png|left|200px]]


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[[Category: Tesmer, J J.]]
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[[Category: Atp-binding]]
[[Category: Inhibitor]]
[[Category: Membrane]]
[[Category: Serine/threonine-protein kinase]]
[[Category: Transferase]]
[[Category: Transferase-signaling protein-inhibitor complex]]

Revision as of 05:14, 27 July 2011

File:3pvu.png

Template:STRUCTURE 3pvu

Bovine GRK2 in complex with Gbetagamma subunits and a selective kinase inhibitor (CMPD101)

Template:ABSTRACT PUBMED 21596927

About this Structure

3pvu is a 3 chain structure with sequence from Bos taurus. Full crystallographic information is available from OCA.

Reference

  1. Thal DM, Yeow RY, Schoenau C, Huber J, Tesmer JJ. Molecular Mechanism of Selectivity Among G Protein-Coupled Receptor Kinase 2 Inhibitors. Mol Pharmacol. 2011 May 19. PMID:21596927 doi:10.1124/mol.111.071522

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