2x0y: Difference between revisions
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[[Image:2x0y.png|left|200px]] | [[Image:2x0y.png|left|200px]] | ||
{{STRUCTURE_2x0y| PDB=2x0y | SCENE= }} | {{STRUCTURE_2x0y| PDB=2x0y | SCENE= }} | ||
===SCREENING-BASED DISCOVERY OF DRUG-LIKE O-GLCNACASE INHIBITOR SCAFFOLDS=== | ===SCREENING-BASED DISCOVERY OF DRUG-LIKE O-GLCNACASE INHIBITOR SCAFFOLDS=== | ||
{{ABSTRACT_PUBMED_20026047}} | {{ABSTRACT_PUBMED_20026047}} | ||
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==See Also== | ==See Also== | ||
*[[Beta-Hexosaminidase]] | *[[Beta-Hexosaminidase|Beta-Hexosaminidase]] | ||
==Reference== | ==Reference== | ||
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[[Category: Aalten, D M.F Van.]] | [[Category: Aalten, D M.F Van.]] | ||
[[Category: Dorfmueller, H C.]] | [[Category: Dorfmueller, H C.]] | ||
[[Category: Cell adhesion]] | |||
[[Category: Glycosidase]] | |||
[[Category: Hydrolase]] | |||
Revision as of 11:23, 25 July 2012
SCREENING-BASED DISCOVERY OF DRUG-LIKE O-GLCNACASE INHIBITOR SCAFFOLDS
Template:ABSTRACT PUBMED 20026047
About this Structure
2x0y is a 2 chain structure of Beta-Hexosaminidase with sequence from Clostridium perfringens. Full crystallographic information is available from OCA.
See Also
Reference
- Dorfmueller HC, van Aalten DM. Screening-based discovery of drug-like O-GlcNAcase inhibitor scaffolds. FEBS Lett. 2010 Feb 19;584(4):694-700. Epub 2009 Dec 16. PMID:20026047 doi:10.1016/j.febslet.2009.12.020