4a7c: Difference between revisions

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[[Image:4a7c.jpg|left|200px]]
[[Image:4a7c.png|left|200px]]


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Revision as of 04:59, 23 May 2012

File:4a7c.png

Template:STRUCTURE 4a7c

Crystal structure of PIM1 kinase with ETP46546

Template:ABSTRACT PUBMED 22266039

About this Structure

4a7c is a 1 chain structure with sequence from Homo sapiens. Full crystallographic information is available from OCA.

Reference

  1. Pastor J, Oyarzabal J, Saluste G, Alvarez RM, Rivero V, Ramos F, Cendon E, Blanco-Aparicio C, Ajenjo N, Cebria A, Albarran MI, Cebrian D, Corrionero A, Fominaya J, Montoya G, Mazzorana M. Hit to lead evaluation of 1,2,3-triazolo[4,5-b]pyridines as PIM kinase inhibitors. Bioorg Med Chem Lett. 2012 Feb 15;22(4):1591-7. Epub 2012 Jan 5. PMID:22266039 doi:10.1016/j.bmcl.2011.12.130

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