1c8k: Difference between revisions
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[[Image:1c8k.gif|left|200px]] | [[Image:1c8k.gif|left|200px]] | ||
'''FLAVOPIRIDOL INHIBITS GLYCOGEN PHOSPHORYLASE BY BINDING AT THE INHIBITOR SITE''' | {{Structure | ||
|PDB= 1c8k |SIZE=350|CAPTION= <scene name='initialview01'>1c8k</scene>, resolution 1.76Å | |||
|SITE= | |||
|LIGAND= <scene name='pdbligand=PLP:PYRIDOXAL-5'-PHOSPHATE'>PLP</scene> and <scene name='pdbligand=CPB:2-(2-CHLORO-PHENYL)-5,7-DIHYDROXY-8-(3-HYDROXY-1-METHYL-PIPERIDIN-4-YL)-4H-BENZOPYRAN-4-ONE'>CPB</scene> | |||
|ACTIVITY= [http://en.wikipedia.org/wiki/Phosphorylase Phosphorylase], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=2.4.1.1 2.4.1.1] | |||
|GENE= | |||
}} | |||
'''FLAVOPIRIDOL INHIBITS GLYCOGEN PHOSPHORYLASE BY BINDING AT THE INHIBITOR SITE''' | |||
==Overview== | ==Overview== | ||
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==About this Structure== | ==About this Structure== | ||
1C8K is a [ | 1C8K is a [[Single protein]] structure of sequence from [http://en.wikipedia.org/wiki/Oryctolagus_cuniculus Oryctolagus cuniculus]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=1C8K OCA]. | ||
==Reference== | ==Reference== | ||
Flavopiridol inhibits glycogen phosphorylase by binding at the inhibitor site., Oikonomakos NG, Schnier JB, Zographos SE, Skamnaki VT, Tsitsanou KE, Johnson LN, J Biol Chem. 2000 Nov 3;275(44):34566-73. PMID:[http:// | Flavopiridol inhibits glycogen phosphorylase by binding at the inhibitor site., Oikonomakos NG, Schnier JB, Zographos SE, Skamnaki VT, Tsitsanou KE, Johnson LN, J Biol Chem. 2000 Nov 3;275(44):34566-73. PMID:[http://www.ncbi.nlm.nih.gov/pubmed/10924512 10924512] | ||
[[Category: Oryctolagus cuniculus]] | [[Category: Oryctolagus cuniculus]] | ||
[[Category: Phosphorylase]] | [[Category: Phosphorylase]] | ||
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[[Category: transferase]] | [[Category: transferase]] | ||
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