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[[Image:4bbm.jpg|left|200px]]
==CRYSTAL STRUCTURE OF THE HUMAN CDKL2 KINASE DOMAIN WITH BOUND TCS 2312==
 
<StructureSection load='4bbm' size='340' side='right' caption='[[4bbm]], [[Resolution|resolution]] 2.00&Aring;' scene=''>
{{STRUCTURE_4bbm|  PDB=4bbm  |  SCENE=  }}
== Structural highlights ==
 
<table><tr><td colspan='2'>[[4bbm]] is a 2 chain structure with sequence from [http://en.wikipedia.org/wiki/Homo_sapiens Homo sapiens]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=4BBM OCA]. For a <b>guided tour on the structure components</b> use [http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=4BBM FirstGlance]. <br>
===CRYSTAL STRUCTURE OF THE HUMAN CDKL2 KINASE DOMAIN WITH BOUND TCS 2312===
</td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=CL:CHLORIDE+ION'>CL</scene>, <scene name='pdbligand=EDO:1,2-ETHANEDIOL'>EDO</scene>, <scene name='pdbligand=TC0:4-[5-[[3-[(CYCLOPROPYLAMINO)METHYL]PHENYL]AMINO]-1H-PYRAZOL-3-YL]-[1,1-BIPHENYL]-2,4-DIOL'>TC0</scene></td></tr>
 
<tr id='related'><td class="sblockLbl"><b>[[Related_structure|Related:]]</b></td><td class="sblockDat">[[4aaa|4aaa]]</td></tr>
 
<tr id='activity'><td class="sblockLbl"><b>Activity:</b></td><td class="sblockDat"><span class='plainlinks'>[http://en.wikipedia.org/wiki/Cyclin-dependent_kinase Cyclin-dependent kinase], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=2.7.11.22 2.7.11.22] </span></td></tr>
==About this Structure==
<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=4bbm FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=4bbm OCA], [http://www.rcsb.org/pdb/explore.do?structureId=4bbm RCSB], [http://www.ebi.ac.uk/pdbsum/4bbm PDBsum]</span></td></tr>
[[4bbm]] is a 2 chain structure with sequence from [http://en.wikipedia.org/wiki/Homo_sapiens Homo sapiens]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=4BBM OCA].  
</table>
__TOC__
</StructureSection>
[[Category: Cyclin-dependent kinase]]
[[Category: Cyclin-dependent kinase]]
[[Category: Homo sapiens]]
[[Category: Homo sapiens]]
[[Category: Arrowsmith, C H.]]
[[Category: Arrowsmith, C H]]
[[Category: Berridge, G.]]
[[Category: Berridge, G]]
[[Category: Bountra, C.]]
[[Category: Bountra, C]]
[[Category: Bullock, A.]]
[[Category: Bullock, A]]
[[Category: Burgess-Brown, N.]]
[[Category: Burgess-Brown, N]]
[[Category: Canning, P.]]
[[Category: Canning, P]]
[[Category: Cooper, C D.O.]]
[[Category: Cooper, C D.O]]
[[Category: Daga, N.]]
[[Category: Daga, N]]
[[Category: Delft, F Von.]]
[[Category: Delft, F Von]]
[[Category: Edwards, A M.]]
[[Category: Edwards, A M]]
[[Category: Elkins, J M.]]
[[Category: Elkins, J M]]
[[Category: Krojer, T.]]
[[Category: Krojer, T]]
[[Category: Mahajan, P.]]
[[Category: Mahajan, P]]
[[Category: Muniz, J R.C.]]
[[Category: Muniz, J R.C]]
[[Category: Phospho-mimetic]]
[[Category: Phospho-mimetic]]
[[Category: Transferase]]
[[Category: Transferase]]

Revision as of 13:29, 4 January 2015

CRYSTAL STRUCTURE OF THE HUMAN CDKL2 KINASE DOMAIN WITH BOUND TCS 2312

4bbm, resolution 2.00Å

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