5aau: Difference between revisions

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==Optimization of a novel binding motif to to (E)-3-(3,5-difluoro-4-((1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-2,3,4,9-tetrahydro-1H- pyrido(3,4-b)indol-1-yl)phenyl)acrylic acid (AZD9496), a potent and orally bioavailable selective estrogen receptor downregulator and antagonist==
==Optimization of a novel binding motif to to (E)-3-(3,5-difluoro-4-((1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-2,3,4,9-tetrahydro-1H- pyrido(3,4-b)indol-1-yl)phenyl)acrylic acid (AZD9496), a potent and orally bioavailable selective estrogen receptor downregulator and antagonist==
<StructureSection load='5aau' size='340' side='right' caption='[[5aau]], [[Resolution|resolution]] 1.90&Aring;' scene=''>
<StructureSection load='5aau' size='340' side='right' caption='[[5aau]], [[Resolution|resolution]] 1.90&Aring;' scene=''>
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</td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=XBR:3-(1-(4-CHLOROPHENYL)-3,4-DIHYDRO-1H-PYRIDO(3,4-B)INDOL-2(9H)-YL)PROPANOIC+ACID'>XBR</scene></td></tr>
</td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=XBR:3-(1-(4-CHLOROPHENYL)-3,4-DIHYDRO-1H-PYRIDO(3,4-B)INDOL-2(9H)-YL)PROPANOIC+ACID'>XBR</scene></td></tr>
<tr id='related'><td class="sblockLbl"><b>[[Related_structure|Related:]]</b></td><td class="sblockDat">[[5aav|5aav]]</td></tr>
<tr id='related'><td class="sblockLbl"><b>[[Related_structure|Related:]]</b></td><td class="sblockDat">[[5aav|5aav]]</td></tr>
<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=5aau FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=5aau OCA], [http://pdbe.org/5aau PDBe], [http://www.rcsb.org/pdb/explore.do?structureId=5aau RCSB], [http://www.ebi.ac.uk/pdbsum/5aau PDBsum]</span></td></tr>
<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=5aau FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=5aau OCA], [http://pdbe.org/5aau PDBe], [http://www.rcsb.org/pdb/explore.do?structureId=5aau RCSB], [http://www.ebi.ac.uk/pdbsum/5aau PDBsum], [http://prosat.h-its.org/prosat/prosatexe?pdbcode=5aau ProSAT]</span></td></tr>
</table>
</table>
== Function ==
== Function ==
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