4rj3: Difference between revisions
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==CDK2 with EGFR inhibitor compound 8== | ==CDK2 with EGFR inhibitor compound 8== | ||
<StructureSection load='4rj3' size='340' side='right' caption='[[4rj3]], [[Resolution|resolution]] 1.63Å' scene=''> | <StructureSection load='4rj3' size='340' side='right'caption='[[4rj3]], [[Resolution|resolution]] 1.63Å' scene=''> | ||
== Structural highlights == | == Structural highlights == | ||
<table><tr><td colspan='2'>[[4rj3]] is a 1 chain structure. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=4RJ3 OCA]. For a <b>guided tour on the structure components</b> use [http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=4RJ3 FirstGlance]. <br> | <table><tr><td colspan='2'>[[4rj3]] is a 1 chain structure with sequence from [http://en.wikipedia.org/wiki/Human Human]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=4RJ3 OCA]. For a <b>guided tour on the structure components</b> use [http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=4RJ3 FirstGlance]. <br> | ||
</td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=3QS:1-CYCLOPENTYL-N-[2-(4-METHOXYPIPERIDIN-1-YL)PYRIMIDIN-4-YL]-1H-PYRROLO[3,2-C]PYRIDIN-6-AMINE'>3QS</scene>, <scene name='pdbligand=ACT:ACETATE+ION'>ACT</scene></td></tr> | </td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=3QS:1-CYCLOPENTYL-N-[2-(4-METHOXYPIPERIDIN-1-YL)PYRIMIDIN-4-YL]-1H-PYRROLO[3,2-C]PYRIDIN-6-AMINE'>3QS</scene>, <scene name='pdbligand=ACT:ACETATE+ION'>ACT</scene></td></tr> | ||
<tr id='NonStdRes'><td class="sblockLbl"><b>[[Non-Standard_Residue|NonStd Res:]]</b></td><td class="sblockDat"><scene name='pdbligand=ALY:N(6)-ACETYLLYSINE'>ALY</scene></td></tr> | <tr id='NonStdRes'><td class="sblockLbl"><b>[[Non-Standard_Residue|NonStd Res:]]</b></td><td class="sblockDat"><scene name='pdbligand=ALY:N(6)-ACETYLLYSINE'>ALY</scene></td></tr> | ||
<tr id='related'><td class="sblockLbl"><b>[[Related_structure|Related:]]</b></td><td class="sblockDat">[[4rj4|4rj4]], [[4rj5|4rj5]], [[4rj6|4rj6]], [[4rj7|4rj7]], [[4rj8|4rj8]]</td></tr> | <tr id='related'><td class="sblockLbl"><b>[[Related_structure|Related:]]</b></td><td class="sblockDat">[[4rj4|4rj4]], [[4rj5|4rj5]], [[4rj6|4rj6]], [[4rj7|4rj7]], [[4rj8|4rj8]]</td></tr> | ||
<tr id='gene'><td class="sblockLbl"><b>[[Gene|Gene:]]</b></td><td class="sblockDat">CDK2, CDKN2 ([http://www.ncbi.nlm.nih.gov/Taxonomy/Browser/wwwtax.cgi?mode=Info&srchmode=5&id=9606 HUMAN])</td></tr> | |||
<tr id='activity'><td class="sblockLbl"><b>Activity:</b></td><td class="sblockDat"><span class='plainlinks'>[http://en.wikipedia.org/wiki/Cyclin-dependent_kinase Cyclin-dependent kinase], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=2.7.11.22 2.7.11.22] </span></td></tr> | <tr id='activity'><td class="sblockLbl"><b>Activity:</b></td><td class="sblockDat"><span class='plainlinks'>[http://en.wikipedia.org/wiki/Cyclin-dependent_kinase Cyclin-dependent kinase], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=2.7.11.22 2.7.11.22] </span></td></tr> | ||
<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=4rj3 FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=4rj3 OCA], [http://pdbe.org/4rj3 PDBe], [http://www.rcsb.org/pdb/explore.do?structureId=4rj3 RCSB], [http://www.ebi.ac.uk/pdbsum/4rj3 PDBsum], [http://prosat.h-its.org/prosat/prosatexe?pdbcode=4rj3 ProSAT]</span></td></tr> | <tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=4rj3 FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=4rj3 OCA], [http://pdbe.org/4rj3 PDBe], [http://www.rcsb.org/pdb/explore.do?structureId=4rj3 RCSB], [http://www.ebi.ac.uk/pdbsum/4rj3 PDBsum], [http://prosat.h-its.org/prosat/prosatexe?pdbcode=4rj3 ProSAT]</span></td></tr> | ||
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</StructureSection> | </StructureSection> | ||
[[Category: Cyclin-dependent kinase]] | [[Category: Cyclin-dependent kinase]] | ||
[[Category: Human]] | |||
[[Category: Large Structures]] | |||
[[Category: Eigenbrot, C]] | [[Category: Eigenbrot, C]] | ||
[[Category: Yin, J]] | [[Category: Yin, J]] | ||