2vip: Difference between revisions

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[[Image:2vip.jpg|left|200px]]
[[Image:2vip.jpg|left|200px]]


{{Structure
<!--
|PDB= 2vip |SIZE=350|CAPTION= <scene name='initialview01'>2vip</scene>, resolution 1.72&Aring;
The line below this paragraph, containing "STRUCTURE_2vip", creates the "Structure Box" on the page.
|SITE= <scene name='pdbsite=AC1:Act+Binding+Site+For+Chain+A'>AC1</scene>, <scene name='pdbsite=AC2:So4+Binding+Site+For+Chain+A'>AC2</scene> and <scene name='pdbsite=AC3:L1r+Binding+Site+For+Chain+A'>AC3</scene>
You may change the PDB parameter (which sets the PDB file loaded into the applet)  
|LIGAND= <scene name='pdbligand=ACT:ACETATE+ION'>ACT</scene>, <scene name='pdbligand=L1R:4-(2-AMINOETHOXY)-3,5-DICHLORO-N-[3-(1-METHYLETHOXY)PHENYL]BENZAMIDE'>L1R</scene>, <scene name='pdbligand=SO4:SULFATE+ION'>SO4</scene>
or the SCENE parameter (which sets the initial scene displayed when the page is loaded),
|ACTIVITY= <span class='plainlinks'>[http://en.wikipedia.org/wiki/U-plasminogen_activator U-plasminogen activator], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=3.4.21.73 3.4.21.73] </span>
or leave the SCENE parameter empty for the default display.
|GENE=  
-->
|DOMAIN=
{{STRUCTURE_2vip| PDB=2vip  | SCENE= }}  
|RELATEDENTRY=[[2viv|2VIV]], [[1c5x|1C5X]], [[1gj9|1GJ9]], [[2vio|2VIO]], [[1w0z|1W0Z]], [[1fv9|1FV9]], [[1vja|1VJA]], [[1gj8|1GJ8]], [[1w11|1W11]], [[1sqo|1SQO]], [[1gjd|1GJD]], [[1w10|1W10]], [[1owk|1OWK]], [[1w12|1W12]], [[1gi9|1GI9]], [[1o5a|1O5A]], [[1c5z|1C5Z]], [[1owj|1OWJ]], [[1gi7|1GI7]], [[1o5b|1O5B]], [[1gjc|1GJC]], [[1sc8|1SC8]], [[1gja|1GJA]], [[1o3p|1O3P]], [[1owe|1OWE]], [[1sqa|1SQA]], [[1gjb|1GJB]], [[2viw|2VIW]], [[1f92|1F92]], [[1owi|1OWI]], [[1kdu|1KDU]], [[2vin|2VIN]], [[1sqt|1SQT]], [[1f5l|1F5L]], [[1owd|1OWD]], [[1ejn|1EJN]], [[2viq|2VIQ]], [[1lmw|1LMW]], [[1u6q|1U6Q]], [[1gi8|1GI8]], [[2jde|2JDE]], [[1c5y|1C5Y]], [[1w14|1W14]], [[1vj9|1VJ9]], [[1w13|1W13]], [[1gj7|1GJ7]], [[1c5w|1C5W]], [[1owh|1OWH]], [[1o5c|1O5C]]
|RESOURCES=<span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=2vip FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=2vip OCA], [http://www.ebi.ac.uk/pdbsum/2vip PDBsum], [http://www.rcsb.org/pdb/explore.do?structureId=2vip RCSB]</span>
}}


'''FRAGMENT-BASED DISCOVERY OF MEXILETINE DERIVATIVES AS ORALLY BIOAVAILABLE INHIBITORS OF UROKINASE-TYPE PLASMINOGEN ACTIVATOR'''
'''FRAGMENT-BASED DISCOVERY OF MEXILETINE DERIVATIVES AS ORALLY BIOAVAILABLE INHIBITORS OF UROKINASE-TYPE PLASMINOGEN ACTIVATOR'''
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[[Category: Vinkovic, M.]]
[[Category: Vinkovic, M.]]
[[Category: Wallis, N G.]]
[[Category: Wallis, N G.]]
[[Category: blood coagulation]]
[[Category: Blood coagulation]]
[[Category: egf-like domain]]
[[Category: Egf-like domain]]
[[Category: fibrinolysis]]
[[Category: Fibrinolysis]]
[[Category: glycoprotein]]
[[Category: Glycoprotein]]
[[Category: hydrolase]]
[[Category: Hydrolase]]
[[Category: inhibitor]]
[[Category: Inhibitor]]
[[Category: kringle]]
[[Category: Kringle]]
[[Category: pharmaceutical]]
[[Category: Pharmaceutical]]
[[Category: phosphorylation]]
[[Category: Phosphorylation]]
[[Category: plasminogen activation]]
[[Category: Plasminogen activation]]
[[Category: polymorphism]]
[[Category: Polymorphism]]
[[Category: protease]]
[[Category: Protease]]
[[Category: secreted]]
[[Category: Secreted]]
[[Category: serine protease]]
[[Category: Serine protease]]
[[Category: urokinase-type plasminogen activator]]
[[Category: Urokinase-type plasminogen activator]]
[[Category: zymogen]]
[[Category: Zymogen]]
 
''Page seeded by [http://oca.weizmann.ac.il/oca OCA ] on Sun May  4 18:52:57 2008''
''Page seeded by [http://oca.weizmann.ac.il/oca OCA ] on Mon Mar 31 05:12:47 2008''