PROTAC: Difference between revisions

From Proteopedia
Jump to navigationJump to search
Jaime Prilusky (talk | contribs)
No edit summary
Jaime Prilusky (talk | contribs)
No edit summary
Line 1: Line 1:
PROTAC (proteolysis-targeting chimera) is a small protein with two active domains joined by a linker.
PROTAC (Proteolysis-Targeting Chimera) is a small protein with two active domains joined by a linker.
[[Image:PROTAC_70.png|thumb|right|300px|Representative PROTAC from [https://protacpedia.weizmann.ac.il/ptcb/detp?i=70 PROTACpedia] targeting EGFR Epidermal growth factor receptor P00533. <span class="bg-lightblue"><b>target binding ligand</b></span><span class="bg-lightmagenta"><b>linker</b></span><span class="bg-lightgreen"><b>E3 binder</b></span>]]
[[Image:PROTAC_70.png|thumb|right|300px|Representative PROTAC from [https://protacpedia.weizmann.ac.il/ptcb/detp?i=70 PROTACpedia] targeting EGFR Epidermal growth factor receptor P00533. <span class="bg-lightblue"><b>target binding ligand</b></span><span class="bg-lightmagenta"><b>linker</b></span><span class="bg-lightgreen"><b>E3 binder</b></span>]]