9b9y: Difference between revisions
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==Structural mechanism of CB1R binding to peripheral and biased inverse agonists== | |||
<StructureSection load='9b9y' size='340' side='right'caption='[[9b9y]], [[Resolution|resolution]] 3.50Å' scene=''> | |||
== Structural highlights == | |||
<table><tr><td colspan='2'>[[9b9y]] is a 2 chain structure with sequence from [https://en.wikipedia.org/wiki/Homo_sapiens Homo sapiens], [https://en.wikipedia.org/wiki/Lama_glama Lama glama] and [https://en.wikipedia.org/wiki/Pyrococcus_abyssi_GE5 Pyrococcus abyssi GE5]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=9B9Y OCA]. For a <b>guided tour on the structure components</b> use [https://proteopedia.org/fgij/fg.htm?mol=9B9Y FirstGlance]. <br> | |||
</td></tr><tr id='method'><td class="sblockLbl"><b>[[Empirical_models|Method:]]</b></td><td class="sblockDat" id="methodDat">Electron Microscopy, [[Resolution|Resolution]] 3.5Å</td></tr> | |||
[[Category: | <tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat" id="ligandDat"><scene name='pdbligand=7DY:N-[(2S,3S)-4-(4-CHLOROPHENYL)-3-(3-CYANOPHENYL)BUTAN-2-YL]-2-METHYL-2-{[5-(TRIFLUOROMETHYL)PYRIDIN-2-YL]OXY}PROPANAMIDE'>7DY</scene></td></tr> | ||
<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[https://proteopedia.org/fgij/fg.htm?mol=9b9y FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=9b9y OCA], [https://pdbe.org/9b9y PDBe], [https://www.rcsb.org/pdb/explore.do?structureId=9b9y RCSB], [https://www.ebi.ac.uk/pdbsum/9b9y PDBsum], [https://prosat.h-its.org/prosat/prosatexe?pdbcode=9b9y ProSAT]</span></td></tr> | |||
</table> | |||
__TOC__ | |||
</StructureSection> | |||
[[Category: Homo sapiens]] | |||
[[Category: Lama glama]] | |||
[[Category: Large Structures]] | |||
[[Category: Pyrococcus abyssi GE5]] | |||
[[Category: Enos MD]] | |||
[[Category: Hassan SA]] | |||
[[Category: Iyer MR]] | |||
[[Category: Kumari P]] | |||
[[Category: Kunos G]] | |||
[[Category: Lim D]] | |||
[[Category: Ramesh K]] | |||
[[Category: Rosenbaum DM]] | |||
[[Category: Szabolcs D]] | |||