9ftn: Difference between revisions

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'''Unreleased structure'''


The entry 9ftn is ON HOLD  until Paper Publication
==Crystal Structure of Autotaxin (ENPP2) with Type VI Inhibitor, a Novel Class of Inhibitors with Three-Point Lock Binding Mode==
 
<StructureSection load='9ftn' size='340' side='right'caption='[[9ftn]], [[Resolution|resolution]] 2.90&Aring;' scene=''>
Authors: Borza, R., Joosten, R.P., Perrakis, A.
== Structural highlights ==
 
<table><tr><td colspan='2'>[[9ftn]] is a 1 chain structure with sequence from [https://en.wikipedia.org/wiki/Rattus_norvegicus Rattus norvegicus]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=9FTN OCA]. For a <b>guided tour on the structure components</b> use [https://proteopedia.org/fgij/fg.htm?mol=9FTN FirstGlance]. <br>
Description: Crystal Structure of Autotaxin (ENPP2) with Type VI Inhibitor, a Novel Class of Inhibitors with Three-Point Lock Binding Mode
</td></tr><tr id='method'><td class="sblockLbl"><b>[[Empirical_models|Method:]]</b></td><td class="sblockDat" id="methodDat">X-ray diffraction, [[Resolution|Resolution]] 2.9&#8491;</td></tr>
[[Category: Unreleased Structures]]
<tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat" id="ligandDat"><scene name='pdbligand=A1IG5:3-[3-[[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-methyl-amino]-6-(1-methylsulfonylpiperidin-4-yl)imidazo[1,2-b]pyridazin-2-yl]-~{N}-(2-oxidanylidene-3~{H}-1,3-benzoxazol-6-yl)propanamide'>A1IG5</scene>, <scene name='pdbligand=BMA:BETA-D-MANNOSE'>BMA</scene>, <scene name='pdbligand=CA:CALCIUM+ION'>CA</scene>, <scene name='pdbligand=IOD:IODIDE+ION'>IOD</scene>, <scene name='pdbligand=MAN:ALPHA-D-MANNOSE'>MAN</scene>, <scene name='pdbligand=NAG:N-ACETYL-D-GLUCOSAMINE'>NAG</scene>, <scene name='pdbligand=SCN:THIOCYANATE+ION'>SCN</scene>, <scene name='pdbligand=ZN:ZINC+ION'>ZN</scene></td></tr>
[[Category: Borza, R]]
<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[https://proteopedia.org/fgij/fg.htm?mol=9ftn FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=9ftn OCA], [https://pdbe.org/9ftn PDBe], [https://www.rcsb.org/pdb/explore.do?structureId=9ftn RCSB], [https://www.ebi.ac.uk/pdbsum/9ftn PDBsum], [https://prosat.h-its.org/prosat/prosatexe?pdbcode=9ftn ProSAT]</span></td></tr>
[[Category: Joosten, R.P]]
</table>
[[Category: Perrakis, A]]
== Function ==
[https://www.uniprot.org/uniprot/ENPP2_RAT ENPP2_RAT]
__TOC__
</StructureSection>
[[Category: Large Structures]]
[[Category: Rattus norvegicus]]
[[Category: Borza R]]
[[Category: Joosten RP]]
[[Category: Perrakis A]]