3qcs: Difference between revisions

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[[Image:3qcs.jpg|left|200px]]
[[Image:3qcs.png|left|200px]]


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Revision as of 07:33, 30 March 2011

File:3qcs.png

Template:STRUCTURE 3qcs

Phosphoinositide-Dependent Kinase-1 (PDK1) kinase domain with 6-[2-Amino-6-(4-morpholinyl)-4-pyrimidinyl]-1H-indazol-3-amine

Template:ABSTRACT PUBMED 21341675

About this Structure

3qcs is a 1 chain structure with sequence from Homo sapiens. Full crystallographic information is available from OCA.

Reference

  1. Medina JR, Becker CJ, Blackledge CW, Duquenne C, Feng Y, Grant SW, Heerding D, Li WH, Miller WH, Romeril SP, Scherzer D, Shu A, Bobko MA, Chadderton AR, Dumble M, Gardiner CM, Gilbert S, Liu Q, Rabindran SK, Sudakin V, Xiang H, Brady PG, Campobasso N, Ward P, Axten JM. Structure-Based Design of Potent and Selective 3-Phosphoinositide-Dependent Kinase-1 (PDK1) Inhibitors. J Med Chem. 2011 Feb 22. PMID:21341675 doi:10.1021/jm101527u

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