Sandbox 121: Difference between revisions
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Notable differences between carazolol and both isoproterenol and the natural agonist norepinephrine are that: | Notable differences between carazolol and both isoproterenol and the natural agonist norepinephrine are that: | ||
(i) Carazolol lacks the hydroxyl groups thought to be necessary for the activation of β₂AR. | (i) Carazolol lacks the hydroxyl groups thought to be necessary for the activation of β₂AR. | ||
(ii) | (ii)The side chain of carazolol is two atoms (one carbon and one oxygen) longer in length from the amino group to the carbazole moiety. | ||
These are common characteristics of β₂AR antagonists. | These are common characteristics of β₂AR antagonists. | ||