4dfu: Difference between revisions

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[[Image:4dfu.jpg|left|200px]]
[[Image:4dfu.png|left|200px]]


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[[Category: Minasov, G.]]
[[Category: Minasov, G.]]
[[Category: Savchenko, A.]]
[[Category: Savchenko, A.]]
[[Category: Shakya, T.]]
[[Category: Stogios, P J.]]
[[Category: Stogios, P J.]]
[[Category: Wright, G D.]]
[[Category: Aminoglycoside phosphotransferase]]
[[Category: Aminoglycoside phosphotransferase]]
[[Category: Aminoglycoside]]
[[Category: Aminoglycoside]]

Revision as of 06:54, 22 February 2012

File:4dfu.png

Template:STRUCTURE 4dfu

Inhibition of an antibiotic resistance enzyme: crystal structure of aminoglycoside phosphotransferase APH(2")-ID/APH(2")-IVA in complex with kanamycin inhibited with quercetin

Template:ABSTRACT PUBMED 22195561

About this Structure

4dfu is a 2 chain structure with sequence from Enterococcus casseliflavus and Streptomyces kanamyceticus. This structure supersedes the now removed PDB entries and 3r82. Full crystallographic information is available from OCA.

Reference

  1. Shakya T, Stogios PJ, Waglechner N, Evdokimova E, Ejim L, Blanchard JE, McArthur AG, Savchenko A, Wright GD. A small molecule discrimination map of the antibiotic resistance kinome. Chem Biol. 2011 Dec 23;18(12):1591-601. PMID:22195561 doi:10.1016/j.chembiol.2011.10.018

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