2bsm: Difference between revisions
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[[Image:2bsm.png|left|200px]] | [[Image:2bsm.png|left|200px]] | ||
{{STRUCTURE_2bsm| PDB=2bsm | SCENE= }} | {{STRUCTURE_2bsm| PDB=2bsm | SCENE= }} | ||
===NOVEL, POTENT SMALL MOLECULE INHIBITORS OF THE MOLECULAR CHAPERONE HSP90 DISCOVERED THROUGH STRUCTURE-BASED DESIGN=== | ===NOVEL, POTENT SMALL MOLECULE INHIBITORS OF THE MOLECULAR CHAPERONE HSP90 DISCOVERED THROUGH STRUCTURE-BASED DESIGN=== | ||
{{ABSTRACT_PUBMED_15974572}} | {{ABSTRACT_PUBMED_15974572}} | ||
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==See Also== | ==See Also== | ||
*[[Heat Shock Proteins]] | *[[Heat Shock Proteins|Heat Shock Proteins]] | ||
==Reference== | ==Reference== | ||
<ref group="xtra">PMID: | <ref group="xtra">PMID:015974572</ref><references group="xtra"/> | ||
[[Category: Homo sapiens]] | [[Category: Homo sapiens]] | ||
[[Category: Barril, X.]] | [[Category: Barril, X.]] | ||
Revision as of 22:05, 26 July 2012
NOVEL, POTENT SMALL MOLECULE INHIBITORS OF THE MOLECULAR CHAPERONE HSP90 DISCOVERED THROUGH STRUCTURE-BASED DESIGN
Template:ABSTRACT PUBMED 15974572
About this Structure
2bsm is a 1 chain structure of Heat Shock Proteins with sequence from Homo sapiens. Full crystallographic information is available from OCA.
See Also
Reference
- Dymock BW, Barril X, Brough PA, Cansfield JE, Massey A, McDonald E, Hubbard RE, Surgenor A, Roughley SD, Webb P, Workman P, Wright L, Drysdale MJ. Novel, potent small-molecule inhibitors of the molecular chaperone Hsp90 discovered through structure-based design. J Med Chem. 2005 Jun 30;48(13):4212-5. PMID:15974572 doi:10.1021/jm050355z