2wip: Difference between revisions
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{{STRUCTURE_2wip| PDB=2wip | SCENE= }} | {{STRUCTURE_2wip| PDB=2wip | SCENE= }} | ||
===STRUCTURE OF CDK2-CYCLIN A COMPLEXED WITH 8-ANILINO-1-METHYL-4,5-DIHYDRO-1H-PYRAZOLO[4,3-H] QUINAZOLINE-3-CARBOXYLIC ACID=== | ===STRUCTURE OF CDK2-CYCLIN A COMPLEXED WITH 8-ANILINO-1-METHYL-4,5-DIHYDRO- 1H-PYRAZOLO[4,3-H] QUINAZOLINE-3-CARBOXYLIC ACID=== | ||
{{ABSTRACT_PUBMED_19603809}} | {{ABSTRACT_PUBMED_19603809}} | ||
==About this Structure== | ==About this Structure== | ||
[[2wip]] is a 4 chain structure of [[Cell Division Protein Kinase 2]] and [[Cyclin] | [[2wip]] is a 4 chain structure of [[Cell Division Protein Kinase 2]] and [[Cyclin]]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=2WIP OCA]. | ||
==See Also== | ==See Also== | ||
| Line 16: | Line 16: | ||
==Reference== | ==Reference== | ||
<ref group="xtra">PMID:019603809</ref><references group="xtra"/> | <ref group="xtra">PMID:019603809</ref><references group="xtra"/> | ||
[[Category: Non-specific serine/threonine protein kinase]] | [[Category: Non-specific serine/threonine protein kinase]] | ||
[[Category: Amboldi, N.]] | [[Category: Amboldi, N.]] | ||
Revision as of 06:31, 10 October 2012
STRUCTURE OF CDK2-CYCLIN A COMPLEXED WITH 8-ANILINO-1-METHYL-4,5-DIHYDRO- 1H-PYRAZOLO[4,3-H] QUINAZOLINE-3-CARBOXYLIC ACID
Template:ABSTRACT PUBMED 19603809
About this Structure
2wip is a 4 chain structure of Cell Division Protein Kinase 2 and Cyclin. Full crystallographic information is available from OCA.
See Also
Reference
- Brasca MG, Amboldi N, Ballinari D, Cameron A, Casale E, Cervi G, Colombo M, Colotta F, Croci V, D'Alessio R, Fiorentini F, Isacchi A, Mercurio C, Moretti W, Panzeri A, Pastori W, Pevarello P, Quartieri F, Roletto F, Traquandi G, Vianello P, Vulpetti A, Ciomei M. Identification of N,1,4,4-Tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydr o-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide (PHA-848125), a Potent, Orally Available Cyclin Dependent Kinase Inhibitor. J Med Chem. 2009 Jul 15. PMID:19603809 doi:10.1021/jm9006559
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Categories:
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- Non-specific serine/threonine protein kinase
- Amboldi, N.
- Ballinari, D.
- Brasca, M G.
- Cameron, A D.
- Casale, E.
- Cervi, G.
- Ciomei, M.
- Colombo, M.
- Colotta, F.
- Croci, V.
- Dalessio, R.
- Fiorentini, F.
- Isacchi, A.
- Mercurio, C.
- Moretti, W.
- Panzeri, A.
- Pastori, W.
- Pevarello, P.
- Quartieri, F.
- Roletto, F.
- Traquandi, G.
- Vianello, P.
- Vulpetti, A.
- Atp-binding
- Cell cycle
- Cell division
- Cyclin
- Kinase
- Mitosis
- Nucleotide-binding
- Nucleus
- Phosphoprotein
- Phosphorylation
- Protein kinase
- Serine/threonine-protein 2 kinase
- Serine/threonine-protein kinase
- Transferase