4nqn: Difference between revisions

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{{STRUCTURE_4nqn|  PDB=4nqn  |  SCENE=  }}
==Crystal Structure of the bromodomain of human BRD9 in complex with a triazolo-phthalazine ligand==
===Crystal Structure of the bromodomain of human BRD9 in complex with a triazolo-phthalazine ligand===
<StructureSection load='4nqn' size='340' side='right' caption='[[4nqn]], [[Resolution|resolution]] 1.73&Aring;' scene=''>
 
== Structural highlights ==
==About this Structure==
<table><tr><td colspan='2'>[[4nqn]] is a 1 chain structure with sequence from [http://en.wikipedia.org/wiki/Human Human]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=4NQN OCA]. For a <b>guided tour on the structure components</b> use [http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=4NQN FirstGlance]. <br>
[[4nqn]] is a 1 chain structure. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=4NQN OCA].  
</td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=Y1Z:2-CHLORO-N-[5-(3-METHYL[1,2,4]TRIAZOLO[3,4-A]PHTHALAZIN-6-YL)-2-(MORPHOLIN-4-YL)PHENYL]BENZENESULFONAMIDE'>Y1Z</scene></td></tr>
[[Category: Arrowsmith, C H.]]
<tr id='related'><td class="sblockLbl"><b>[[Related_structure|Related:]]</b></td><td class="sblockDat">[[4nqm|4nqm]]</td></tr>
[[Category: Bountra, C.]]
<tr id='gene'><td class="sblockLbl"><b>[[Gene|Gene:]]</b></td><td class="sblockDat">BRD9 ([http://www.ncbi.nlm.nih.gov/Taxonomy/Browser/wwwtax.cgi?mode=Info&srchmode=5&id=9606 HUMAN])</td></tr>
[[Category: Delft, F von.]]
<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=4nqn FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=4nqn OCA], [http://www.rcsb.org/pdb/explore.do?structureId=4nqn RCSB], [http://www.ebi.ac.uk/pdbsum/4nqn PDBsum]</span></td></tr>
[[Category: Edwards, A M.]]
</table>
[[Category: Fedorov, O.]]
__TOC__
[[Category: Felletar, I.]]
</StructureSection>
[[Category: Filippakopoulos, P.]]
[[Category: Human]]
[[Category: Knapp, S.]]
[[Category: Arrowsmith, C H]]
[[Category: Martin, S.]]
[[Category: Bountra, C]]
[[Category: Picaud, S.]]
[[Category: Delft, F von]]
[[Category: SGC, Structural Genomics Consortium.]]
[[Category: Edwards, A M]]
[[Category: Fedorov, O]]
[[Category: Felletar, I]]
[[Category: Filippakopoulos, P]]
[[Category: Knapp, S]]
[[Category: Martin, S]]
[[Category: Picaud, S]]
[[Category: Structural genomic]]
[[Category: Bromodomain]]
[[Category: Bromodomain]]
[[Category: Inhibition]]
[[Category: Inhibition]]
[[Category: Sgc]]
[[Category: Sgc]]
[[Category: Small molecule inhibitor]]
[[Category: Small molecule inhibitor]]
[[Category: Structural genomics consortium]]
[[Category: Transcription]]
[[Category: Transcription]]
[[Category: Transcription-inhibitor complex]]
[[Category: Transcription-inhibitor complex]]