2wih | pdb_00002wih
From Proteopedia
STRUCTURE OF CDK2-CYCLIN A WITH PHA-848125
Template:ABSTRACT PUBMED 19603809
About this Structure
2wih is a 4 chain structure of Cell Division Protein Kinase 2 and Cyclin with sequence from Homo sapiens. Full crystallographic information is available from OCA.
See Also
Reference
- Brasca MG, Amboldi N, Ballinari D, Cameron A, Casale E, Cervi G, Colombo M, Colotta F, Croci V, D'Alessio R, Fiorentini F, Isacchi A, Mercurio C, Moretti W, Panzeri A, Pastori W, Pevarello P, Quartieri F, Roletto F, Traquandi G, Vianello P, Vulpetti A, Ciomei M. Identification of N,1,4,4-Tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydr o-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide (PHA-848125), a Potent, Orally Available Cyclin Dependent Kinase Inhibitor. J Med Chem. 2009 Jul 15. PMID:19603809 doi:10.1021/jm9006559
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Categories:
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- Homo sapiens
- Non-specific serine/threonine protein kinase
- Amboldi, N.
- Ballinari, D.
- Brasca, M G.
- Cameron, A D.
- Casale, E.
- Cervi, G.
- Ciomei, M.
- Colombo, M.
- Colotta, F.
- Croci, V.
- Dalessio, R.
- Fiorentini, F.
- Isacchi, A.
- Mercurio, C.
- Moretti, W.
- Panzeri, A.
- Pastori, W.
- Pevarello, P.
- Quartieri, F.
- Roletto, F.
- Traquandi, G.
- Vianello, P.
- Vulpetti, A.