3u5l | pdb_00003u5l
From Proteopedia
Crystal Structure of the first bromodomain of human BRD4 in complex with a benzo-triazepine ligand (BzT-7)
About this Structure
3u5l is a 1 chain structure with sequence from Homo sapiens. Full crystallographic information is available from OCA.
Reference
- Filippakopoulos P, Picaud S, Fedorov O, Keller M, Wrobel M, Morgenstern O, Bracher F, Knapp S. Benzodiazepines and benzotriazepines as protein interaction inhibitors targeting bromodomains of the BET family. Bioorg Med Chem. 2011 Nov 4. PMID:22137933 doi:10.1016/j.bmc.2011.10.080
Proteopedia Page Contributors and Editors (what is this?)
Categories:
- Pages with broken file links
- Homo sapiens
- Arrowsmith, C H.
- Bountra, C.
- Bracher, F.
- Delft, F von.
- Edwards, A M.
- Fedorov, O.
- Felletar, I.
- Filippakopoulos, P.
- Knapp, S.
- Picaud, S.
- SGC, Structural Genomics Consortium.
- Weigelt, J.
- Brd4
- Bromodomain containing protein 4
- Bromodomain-containing protein 4 isoform long
- Cap
- Hunk1
- Mcap
- Mitotic chromosome associated protein
- Sgc
- Signaling protein-inhibitor complex
- Structural genomics consortium
