3m2w | pdb_00003m2w
From Proteopedia
Crystal structure of MAPKAK kinase 2 (MK2) complexed with a spiroazetidine-tetracyclic ATP site inhibitor
Template:ABSTRACT PUBMED 20591669
About this Structure
3m2w is a 1 chain structure of Mitogen-activated protein kinase with sequence from Homo sapiens. Full crystallographic information is available from OCA.
See Also
Reference
- Revesz L, Schlapbach A, Aichholz R, Dawson J, Feifel R, Hawtin S, Littlewood-Evans A, Koch G, Kroemer M, Mobitz H, Scheufler C, Velcicky J, Huppertz C. In vivo and in vitro SAR of tetracyclic MAPKAP-K2 (MK2) inhibitors. Part II. Bioorg Med Chem Lett. 2010 Aug 1;20(15):4719-23. Epub 2010 Apr 11. PMID:20591669 doi:10.1016/j.bmcl.2010.04.023
Proteopedia Page Contributors and Editors (what is this?)
Categories:
- Pages with broken file links
- Homo sapiens
- Non-specific serine/threonine protein kinase
- Be, C.
- Huppertz, C.
- Izaac, A.
- Kroemer, M.
- Revesz, L.
- Scheufler, C.
- Schlapbach, A.
- Atp-binding
- Atp-site kinase inhibitor
- Kinase
- Novartis compound nvp-bxs169
- Nucleotide-binding
- Phosphoprotein
- Serine/threonine-protein kinase
- Small molecule inhibitor
- Spiroazetidine-tetracycle
- Transferase
