3faa | pdb_00003faa
From Proteopedia
Crystal structure of TGFbRI complexed with a 2-aminoimidazole inhibitor
About this Structure
3faa is a 5 chain structure with sequence from Homo sapiens. Full crystallographic information is available from OCA.
Reference
- Bonafoux D, Chuaqui C, Boriack-Sjodin PA, Fitch C, Hankins G, Josiah S, Black C, Hetu G, Ling L, Lee WC. 2-Aminoimidazoles inhibitors of TGF-beta receptor 1. Bioorg Med Chem Lett. 2009 Feb 1;19(3):912-6. Epub 2008 Dec 11. PMID:19135364 doi:10.1016/j.bmcl.2008.11.119
Proteopedia Page Contributors and Editors (what is this?)
Categories:
- Pages with broken file links
- Homo sapiens
- Receptor protein serine/threonine kinase
- Boriack-Sjodin, P A.
- Fitch, C.
- Atp-binding
- Craniosynostosis
- Disease mutation
- Glycoprotein
- Kinase
- Magnesium
- Manganese
- Membrane
- Metal-binding
- Nucleotide-binding
- Phosphoprotein
- Protein-inhibitor complex
- Receptor
- Serine/threonine-protein kinase
- Structure-based drug design
- Tgfbeta
- Transferase
- Transmembrane