3q9b | pdb_00003q9b

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Template:STRUCTURE 3q9b

Crystal Structure of APAH complexed with M344

Template:ABSTRACT PUBMED 21268586

Function

[APHA_MYCRA] Acts on many types of acetylpolyamines. Has high affinity towards acetylputrescine, acetylcadaverine, acetylspermidine, and acetylspermine. Acts on L-Lys-(epsilon-acetyl)-coumarin, but has very low activity towards acetylated peptides.

About this Structure

3q9b is a 12 chain structure with sequence from Mycoplana ramosa. Full crystallographic information is available from OCA.

Reference

  1. Lombardi PM, Angell HD, Whittington DA, Flynn EF, Rajashankar KR, Christianson DW. Structure of Prokaryotic Polyamine Deacetylase Reveals Evolutionary Functional Relationships with Eukaryotic Histone Deacetylases . Biochemistry. 2011 Jan 26. PMID:21268586 doi:10.1021/bi101859k

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