3kga | pdb_00003kga
From Proteopedia
Crystal structure of MAPKAP kinase 2 (MK2) complexed with a potent 3-aminopyrazole ATP site inhibitor
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Proteopedia Page Contributors and Editors (what is this?)
Categories:
- Homo sapiens
- Non-specific serine/threonine protein kinase
- Be, C.
- Huppertz, C.
- Izaac, A.
- Kroemer, M.
- Pflieger, D.
- Scheufler, C.
- Schlapbach, A.
- Velcicky, J.
- 3-aminopyrazole scaffold
- Activation loop deletion
- Atp-binding
- Atp-site kinase inhibitor
- Induced fit
- Kinase
- Novel hydrophobic pocket
- Nucleotide-binding
- Phosphoprotein
- Scaffold hoping
- Serine/threonine-protein kinase
- Small molecule inhibitor
- Transferase