2q8i | pdb_00002q8i

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Template:STRUCTURE 2q8i

File:2q8i.png

Pyruvate dehydrogenase kinase isoform 3 in complex with antitumor drug radicicol

Template:ABSTRACT PUBMED 17683942

About this Structure

2Q8I is a 2 chains structure of sequences from Homo sapiens. Full crystallographic information is available from OCA.

Reference

  1. Kato M, Li J, Chuang JL, Chuang DT. Distinct structural mechanisms for inhibition of pyruvate dehydrogenase kinase isoforms by AZD7545, dichloroacetate, and radicicol. Structure. 2007 Aug;15(8):992-1004. Epub 2007 Aug 2. PMID:17683942 doi:10.1016/j.str.2007.07.001

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