Telaprevir

From Proteopedia

Telaprevir (VX-950), marketed under the brand names Incivek and Incivo, is a pharmaceutical drug for the treatment of hepatitis C co-developed by Vertex Pharmaceuticals and Johnson & Johnson. It is a member of a class of antiviral drugs known as protease inhibitors. Specifically, telaprevir inhibits the hepatitis C viral enzyme NS3/4A serine protease. See also [1].

Crystal structure of NS3/4A protease in complex with Telaprevir (3sv6).

Telaprevir binding site.

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Crystal structure of NS3/4A protease in complex with Telaprevir (3sv6)

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References

Proteopedia Page Contributors and Editors (what is this?)

Alexander Berchansky

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Telaprevir

From Proteopedia

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